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ACTR2

ACTR2,全稱為肌動蛋白相關蛋白2,是一種參與細胞骨架結構和功能的蛋白。它屬于肌動蛋白相關蛋白家族,與肌動蛋白相互作用,在維持細胞形態、細胞運動和信號傳導中發揮重要作用。ACTR2蛋白也被稱為肌動蛋白相關蛋白A2,是肌動蛋白相關蛋白家族中研究較多的成員之一。
ACTR2主要存在于脂肪和肌肉組織中。在脂肪細胞中,它參與脂質存儲的調控,影響脂肪的合成和分解。在肌肉細胞中,ACTR2蛋白則與肌肉萎縮相關,參與肌肉蛋白的合成和分解,影響肌肉的生長和萎縮。因此,靶向ACTR2蛋白有望在治療肥胖和肌肉萎縮等疾病中發揮作用。
近年來,ACTR2成為藥物研發的熱點靶點。研究表明,抑制ACTR2蛋白的活性可以減少脂肪的合成和儲存,同時促進肌肉蛋白的合成,從而達到減脂增肌的效果。目前,已有多種針對ACTR2蛋白的藥物進入臨床研究階段,包括抗體藥物和融合蛋白等。其中,禮來的Bimagrumab和來凱醫藥的LAE102兩款抗體藥物已率先進入以肥胖為適應癥的臨床研究,并取得了顯著的療效。

熱銷產品

Recombinant Human Actin-related protein 2 (ACTR2) (CSB-EP001248HU)

驗證數據

CSB-EP001248HU

(Tris-Glycine gel) Discontinuous SDS-PAGE (reduced) with 5% enrichment gel and 15% separation gel.

ACTR2 Recombinant Monoclonal Antibody (CSB-RA144588A0HU)

驗證數據

CSB-RA144588A0HU

Western Blot
, Positive WB detected in:Jurkat whole cell lysate(30μg), A549 whole cell lysate(30μg), THP-1 whole cell lysate(30μg), HepG2 whole cell lysate(30μg), MCF7 whole cell lysate(30μg), SH-SY5Y whole cell lysate(30μg), Mouse brain tissue lysate(30μg), Mouse spleen tissue lysate(30μg), Rat kidney lysate(30μg)
All lanes: Actin related protein 2 antibody at 1:1000
Secondary
Goat polyclonal to rabbit IgG at 1/40000 dilution
Predicted band size: 45 kDa
Observed band size: 45 kDa
Exposure time:10s

CSB-RA144588A0HU

Overlay Peak curve showing jurkat cells stained with CSB-RA144588A0HU (red line) at 1:100. The cells were fixed in 4% formaldehyde and permeated by 0.2% TritonX-100 for 10min. Then 10% normal goat serum to block non-specific protein-protein interactions followed by the antibody (1ug/1*106cells) for 45min at 4℃. The secondary antibody used was FITC-conjugated goat anti-rabbit IgG (H+L) at 1/200 dilution for 35min at 4℃.Control antibody (green line) was Rabbit IgG (1ug/1*106cells) used under the same conditions. Acquisition of >10, 000 events was performed.

ACTR2 Antibody (CSB-PA001248ESR1HU)

驗證數據

CSB-PA001248ESR1HU

Western blot
All lanes: Actin-related protein 2 antibody at 3μg/ml
Lane 1: Mouse spleen tissue
Lane 2: Jurkat whole cell lysate
Lane 3: MCF-7 whole cell lysate
Secondary
Goat polyclonal to rabbit IgG at 1/10000 dilution
Predicted band size: 45, 46 kDa
Observed band size: 45 kDa

CSB-PA001248ESR1HU

Immunohistochemistry of paraffin-embedded human tonsil tissue using CSB-PA001248ESR1HU at dilution of 1:100

ACTR2 Antibodies

ACTR2 for Homo sapiens (Human)

ACTR2 Proteins

ACTR2 Proteins for Homo sapiens (Human)